SAR Turns One Hit into a Chemical Series
Structure-activity relationships emerge from testing systematic analogs of a hit, converting a single active molecule into a gradient that guides optimization.
concept
drug-discoverymedicine
Sources
Coursera: *Lead Selection* (Introduction to Drug Hunting > Introduction to Drug Hunting, part 2), 0:03
Coursera: *Lead Selection* (Introduction to Drug Hunting > Introduction to Drug Hunting, part 2), 2:00